2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3111 | Abemaciclib methanesulfonate | abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate) | CDK |
Abemaciclib methanesulfonate (LY2835219) is a specific and effective inhibitor of CDK4(IC50=2 nM) and CDK6(IC50=10 nM). | |||
T2381 | Abemaciclib | CDK4/6 dual inhibitor,LY2835219 | CDK |
Abemaciclib (LY2835219) is a dual inhibitor of CDK4/6 (IC50=2/10 nM) with selectivity and specificity. Abemaciclib has antitumor activity and is used to treat advanced or metastatic breast cancer. |